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Rosiglitazone

E3L044674

Internal ID: BDB044674

Activity data available Local docking-ready structure

Dock with P37231 Dock with Q07869

Structure

/e3_file/ligand_db/generated/BDB044674/BDB044674.sdf

Basic Properties

Compound ID

E3L044674

Internal ID

BDB044674

Molecular formula

C18H19N3O3S

Molecular weight

357.435000

Exact mass

357.114712

XLogP

2.4909

TPSA

71.5300

HBA / HBD

6 / 1

Rotatable bonds

Heavy atoms / rings

25 / 3

Activity summary

EC50 unknown 0.10000000 nM
96 activity record(s) imported

InChIKey

YASAKCUCGLMORW-UHFFFAOYSA-N

SMILES

CN(CCOc1ccc(CC2SC(=O)NC2=O)cc1)c1ccccn1

Aliases

BDBM50030474 (preferred) Rosiglitazone (source_name) BDBM50030474 (source_id)

E3 Relation

E3 UniProt	Gene / protein	Relation type	Ligand role	Direct	Functional	Docking	Source	Evidence
P37231	PPARG;NR1C3 Peroxisome proliferator-activated receptor gamma	reported_binder	bindingdb_reported	Yes	No	low	BindingDB:BDBM50030474	medium ; target=Peroxisome proliferator-activated receptor gamma
Q07869	PPARA;NR1C1;PPAR Peroxisome proliferator-activated receptor alpha	reported_binder	bindingdb_reported	Yes	No	low	BindingDB:BDBM50030474	medium ; target=Peroxisome proliferator-activated receptor alpha; Peroxisome proliferator-activated receptor gamma

Sources and Literature

Source	Source ID	Source URL	Download URL	DOI / PMID
BindingDB	BDBM50030474	Open	-	10.3109/14756360903468171; 10.1016/j.bmcl.2015.04.029; 10.1016/s0960-894x(99)00603-4; 10.1016/j.bmcl.2019.126664; 10.1021/acs.jmedchem.0c01512; 10.7270/Q2571H79; 10.1016/j.ejmech.2022.114927; 10.7270/Q2JS9TG4; 10.1016/j.ejmech.2015.11.030; 10.1016/j.bmc.2016.03.006; 10.1016/j.bmc.2016.11.014; 10.1016/j.bmc.2017.01.015; 10.1016/j.bmcl.2017.04.061; 10.1016/j.bmc.2017.07.015; 10.1016/j.ejmech.2017.07.015; 10.1016/j.bmc.2018.10.033; 10.1016/j.bmcl.2013.09.010; 10.1021/acs.jmedchem.0c01555; 10.1021/acsmedchemlett.1c00715; 10.1016/j.ejmech.2016.12.047; 10.7270/Q2GB282C; 10.7270/Q2Z60TR5; 10.7270/Q21Z438X; 10.1016/j.bmcl.2014.09.053; 10.1016/j.ejmech.2014.10.083; 10.1016/j.ejmech.2014.11.044; 10.1021/acs.jmedchem.5b00849; 10.1016/j.bmc.2016.08.045; 10.1016/j.bmcl.2017.05.037; 10.1021/acs.jmedchem.7b01285; 10.1016/j.bmcl.2018.03.051; 10.1016/j.ejmech.2017.06.006; 10.1016/j.bmc.2018.09.005; 10.1016/j.bmc.2018.09.006; 10.1016/j.ejmech.2017.06.033; 10.1016/j.bmcl.2018.03.010; 10.1021/acs.jmedchem PMID: 20518620; 25978962; 10612594; 31591015; 33423463; 31865018; 36379105; 26708109; 26988801; 27876250; 28117121; 28465099; 28720328; 28735214; 30429097; 24075729; 33142057; 35450368; 28076827; 35714534; 39185622; 25305688; 25462281; 25497132; 26226490; 27591006; 28539218; 29446942; 29615345; 28609708; 30220602; 30241907; 28667876; 29628329; 30199253; 30296685; 23502212; 31268307; 32096640; 32267688; 31629632; 30702885; 27622746; 30996794; 29940464; 33784603; 34455359; 33620196; 35060744; 34818007; 34954593; 35051813; 35089724; 35325635; 28231521; 32339855; 37243609; 38522113; 38185055; 38677560; 38865743; 22364952; 25437304; 26774923
PubChem	CID77999	Open	-

Structure Files

Kind	Format	Status	Docking use	File / link	Preparation note
canonical_2d	SMILES	raw	Docking-ready	CN(CCOc1ccc(CC2SC(=O)NC2=O)cc1)c1ccccn1	keep_bindingdb_unique
generated_3d	SDF	prepared	Docking-ready	public/e3_file/ligand_db/generated/BDB044674/BDB044674.sdf	Generated from canonical SMILES
generated_3d	MOL2	prepared	Docking-ready	public/e3_file/ligand_db/generated/BDB044674/BDB044674.mol2	Generated from canonical SMILES
docking_ready	PDBQT	prepared	Docking-ready	public/e3_file/ligand_db/generated/BDB044674/BDB044674.pdbqt	Generated from canonical SMILES
image	PNG	prepared	Reference	public/e3_file/ligand_db/generated/BDB044674/BDB044674.png	Generated from canonical SMILES
image	SVG	prepared	Reference	public/e3_file/ligand_db/generated/BDB044674/BDB044674.svg	Generated from canonical SMILES

Activity

Target	Source	Assay	Result	Potency	Literature	Records
Peroxisome proliferator-activated receptor alpha Q07869 E3 ligase component	BindingDB:BDBM50030474	EC50	240 nM	Moderate	DOI: 10.1016/j.ejmech.2015.12.049 PMID: 26774923	1
Peroxisome proliferator-activated receptor alpha Q07869 E3 ligase component	BindingDB:BDBM50030474	EC50	10000 nM	Low	DOI: 10.1016/j.ejmech.2017.06.006 PMID: 28609708	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	IC50	112 nM	Moderate	DOI: 10.1016/j.bmc.2018.10.033 PMID: 30429097	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	IC50	76 nM	High	DOI: 10.1016/j.bmcl.2015.04.029 PMID: 25978962	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	IC50	38 nM	High	DOI: 10.1016/j.ejmech.2015.11.030 PMID: 26708109	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	IC50	298 nM	Moderate	DOI: 10.1016/j.bmc.2017.07.015 PMID: 28720328	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	IC50	88 nM	High	DOI: 10.1021/acs.jmedchem.0c01555 PMID: 33142057	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	IC50	159 nM	Moderate	DOI: 10.1016/j.bmcl.2013.09.010 PMID: 24075729	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	IC50	60000 nM	Low	DOI: 10.7270/Q2JS9TG4	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	IC50	10 nM	Very high	DOI: 10.1016/j.bmc.2016.11.014 PMID: 27876250	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	IC50	22000 nM	Low	DOI: 10.1016/j.bmcl.2017.04.061 PMID: 28465099	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	IC50	4400 nM	Low	DOI: 10.1021/acsmedchemlett.1c00715 PMID: 35450368	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	IC50	76 nM	High	DOI: 10.1016/j.bmcl.2019.126664 PMID: 31591015	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	IC50	103 nM	Moderate	DOI: 10.1016/j.ejmech.2017.07.015 PMID: 28735214	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	IC50	7.7 nM	Very high	DOI: 10.1021/acs.jmedchem.0c01555 PMID: 33142057	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	IC50	90 nM	High	DOI: 10.1021/acsmedchemlett.1c00715 PMID: 35450368	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	IC50	10 nM	Very high	DOI: 10.1016/j.bmc.2016.03.006 PMID: 26988801	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	IC50	292 nM	Moderate	DOI: 10.1016/j.bmc.2017.01.015 PMID: 28117121	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	240 nM	Moderate	DOI: 10.1016/j.bmcl.2018.03.051 PMID: 29615345	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	300 nM	Moderate	DOI: 10.1016/j.bmcl.2017.05.037 PMID: 28539218	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	52 nM	High	DOI: 10.1021/acs.jmedchem.7b01285 PMID: 29446942	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	40 nM	High	DOI: 10.1016/j.ejmech.2016.12.047 PMID: 28076827	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	9 nM	Very high	DOI: 10.7270/Q2BC43SK PMID: 28231521	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	260 nM	Moderate	DOI: 10.1016/j.bmc.2016.08.045 PMID: 27591006	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	87 nM	High	DOI: 10.1021/acs.jmedchem.5b00849 PMID: 26226490	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	481 nM	Moderate	DOI: 10.1021/acs.jmedchem.0c01555 PMID: 33142057	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	297 nM	Moderate	DOI: 10.1021/acs.jmedchem.0c01555 PMID: 33142057	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	134 nM	Moderate	DOI: 10.7270/Q2DJ5KQ6 PMID: 35051813	1
Peroxisome proliferator-activated receptor gamma Q07869 E3 ligase component	BindingDB:BDBM50030474	EC50	120 nM	Moderate	DOI: 10.1016/j.bmc.2012.01.028 PMID: 22364952	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	39 nM	High	DOI: 10.1021/acs.jmedchem.8b00835 PMID: 30199253	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	40 nM	High	DOI: 10.1016/j.ejmech.2017.06.033 PMID: 28667876	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	1 nM	Very high	DOI: 10.7270/Q21Z438X	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	4 nM	Very high	DOI: 10.1021/acs.jnatprod.9b00003 PMID: 31268307	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	326 nM	Moderate	DOI: 10.1021/acs.jmedchem.7b01285 PMID: 29446942	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	100 nM	High	DOI: 10.1016/j.ejmech.2018.09.071 PMID: 30296685	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	14 nM	High	DOI: 10.7270/Q2571H79 PMID: 31865018	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	332 nM	Moderate	DOI: 10.1021/acs.jmedchem.7b01285 PMID: 29446942	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	396 nM	Moderate	DOI: 10.1016/j.bmc.2018.09.005 PMID: 30220602	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	18 nM	High	DOI: 10.1021/acs.jmedchem.8b01848 PMID: 30702885	2 source records
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	40 nM	High	DOI: 10.7270/Q23T9N94 PMID: 35325635	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	191500 nM	Low	DOI: 10.1016/j.ejmech.2021.113388 PMID: 33784603	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	10 nM	Very high	DOI: 10.1016/j.ejmech.2013.02.015 PMID: 23502212	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	44000 nM	Low	DOI: 10.7270/Q2GB282C PMID: 35714534	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	120 nM	Moderate	DOI: 10.1016/j.bmc.2012.01.028 PMID: 22364952	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	27 nM	High	DOI: 10.1021/acsmedchemlett.1c00715 PMID: 35450368	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	280 nM	Moderate	DOI: 10.1021/acs.jmedchem.9b01189 PMID: 32096640	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	1100 nM	Low	DOI: 10.1016/j.bmcl.2017.04.061 PMID: 28465099	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	115 nM	Moderate	DOI: 10.1021/acs.jmedchem.9b01786 PMID: 32267688	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	8 nM	Very high	DOI: 10.1016/j.bmc.2018.10.033 PMID: 30429097	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	0.1 nM	Very high	DOI: 10.7270/Q2Q81JRR PMID: 38677560	1
Peroxisome proliferator-activated receptor gamma Q07869 E3 ligase component	BindingDB:BDBM50030474	EC50	1600 nM	Low	DOI: 10.1021/np500234f PMID: 25437304	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	83 nM	High	DOI: 10.1016/j.bmcl.2018.03.010 PMID: 29628329	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	1600 nM	Low	DOI: 10.1021/np500234f PMID: 25437304	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	95 nM	High	DOI: 10.1021/acs.jmedchem.7b01285 PMID: 29446942	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	169 nM	Moderate	DOI: 10.1021/acs.jmedchem.1c02002 PMID: 35060744	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	83 nM	High	DOI: 10.1021/acs.jmedchem.0c02063 PMID: 33620196	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	120 nM	Moderate	DOI: 10.7270/Q2CR5ZFX PMID: 34954593	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	300 nM	Moderate	DOI: 10.7270/Q2Z03DDS PMID: 32339855	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	10 nM	Very high	DOI: 10.1016/j.bmcl.2014.09.053 PMID: 25305688	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	26 nM	High	DOI: 10.7270/Q2GB282C PMID: 35714534	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	89 nM	High	DOI: 10.1016/s0960-894x(99)00603-4 PMID: 10612594	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	259 nM	Moderate	DOI: 10.1016/j.bmcl.2019.126709 PMID: 31629632	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	200 nM	Moderate	DOI: 10.1016/j.ejmech.2018.06.034 PMID: 29940464	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	156 nM	Moderate	DOI: 10.1016/j.ejmech.2021.113807 PMID: 34455359	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	40 nM	High	DOI: 10.1021/acsmedchemlett.8b00574 PMID: 30996794	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	396 nM	Moderate	DOI: 10.1016/j.bmc.2018.09.006 PMID: 30241907	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	39 nM	High	DOI: 10.1016/j.ejmech.2014.10.083 PMID: 25462281	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	155 nM	Moderate	DOI: 10.1021/acs.jmedchem.2c02123 PMID: 37243609	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	730 nM	Moderate	DOI: 10.7270/Q2BC43SK PMID: 28231521	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	49 nM	High	DOI: 10.7270/Q2H99983 PMID: 35089724	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	60 nM	High	DOI: 10.7270/Q2Q244WN PMID: 38185055	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	20 nM	High	DOI: 10.1007/s00044-010-9428-9	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	210 nM	Moderate	DOI: 10.1021/acs.jmedchem.9b01786 PMID: 32267688	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	39 nM	High	DOI: 10.7270/Q2RX9HR7 PMID: 38865743	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	316 nM	Moderate	DOI: 10.1021/acs.jmedchem.7b01285 PMID: 29446942	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	200 nM	Moderate	DOI: 10.7270/Q25X2FHB PMID: 38522113	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	260 nM	Moderate	DOI: 10.1016/j.bmc.2016.08.067 PMID: 27622746	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	76 nM	High	DOI: 10.1021/acs.jmedchem.0c01555 PMID: 33142057	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	40 nM	High	DOI: 10.1016/j.ejmech.2014.11.044 PMID: 25497132	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	4 nM	Very high	DOI: 10.1016/j.ejmech.2017.06.006 PMID: 28609708	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	120 nM	Moderate	DOI: 10.1016/j.ejmech.2018.09.071 PMID: 30296685	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	100 nM	High	DOI: 10.1021/acs.jmedchem.1c01331 PMID: 34818007	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	114 nM	Moderate	DOI: 10.1021/acs.jmedchem.7b01285 PMID: 29446942	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	EC50	117 nM	Moderate	DOI: 10.1021/acs.jmedchem.7b01285 PMID: 29446942	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	Kd	3300 nM	Low	DOI: 10.7270/Q2GB282C PMID: 35714534	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	Kd	1.2 nM	Very high	DOI: 10.1016/j.ejmech.2016.12.047 PMID: 28076827	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	Kd	48 nM	High	DOI: 10.1021/acs.jmedchem.0c01555 PMID: 33142057	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	Kd	3380 nM	Low	DOI: 10.7270/Q2Z60TR5 PMID: 39185622	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	Ki	26 nM	High	DOI: 10.7270/Q2571H79 PMID: 31865018	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	Ki	20 nM	High	DOI: 10.1016/j.ejmech.2022.114927 PMID: 36379105	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	Ki	59 nM	High	DOI: 10.1016/j.bmcl.2019.126664 PMID: 31591015	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	Ki	27 nM	High	DOI: 10.1016/j.bmcl.2015.04.029 PMID: 25978962	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	Ki	8 nM	Very high	DOI: 10.3109/14756360903468171 PMID: 20518620	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	Ki	47 nM	High	DOI: 10.1016/s0960-894x(99)00603-4 PMID: 10612594	1
Peroxisome proliferator-activated receptor gamma P37231 E3 ligase component	BindingDB:BDBM50030474	Ki	17 nM	High	DOI: 10.1021/acs.jmedchem.0c01512 PMID: 33423463	1